Dark spots

How to get rid of hyperpigmentation instantly in 2024

Do you look in the mirror and see dark patches or uneven skin tone?

Maybe you just want to know how to restore that youthful glow.

Either way, you’ve come to the right place.

In this article, we’ll be discussing three critical anti-pigmentation ingredients.

So you can leave this page lighter and brighter than you started.

Three key ingredients

In this series, we have been discussing all things dark spots and pigmentation.

A big question our clients often ask us is how to get rid of hyperpigmentation. This guide outlines the three superhero ingredients that we see excellent results within our clinic:

  • ferulic acid
  • malic acid
  • vitamin C in the form of 3.0 ethyl ascorbic acid

What is hyperpigmentation?

“Hyper” means more, and “pigment” refers to colour.

Hyperpigmentation occurs in your skin when the troublesome enzyme tyrosinase initiates melanin production the pigment responsible for dark spots.

But please don’t be too hard on tyrosinase; it is there to protect you.

Tyrosinase is your skin’s defence mechanism against damage caused by troublesome UV rays, pollution, picking, and scarring.

Whenever your skin is damaged, this enzyme comes to the rescue, flooding the injured area, which is the hyperpigmentation you see in your skin.

So maybe tyrosinase doesn’t deserve the bad rap it gets after all? But boy, can it be challenging to treat.

This article gives a detailed overview if you want to learn more about how to get rid of hyperpigmentation.

How to Get Rid of Hyperpigmentation

It makes sense that targeting this enzyme is the most effective way to control excess melanin production and dark spots on the skin.

It often takes much longer to eliminate pigmentation than to accumulate, especially if you’ve spent years in the sun or dealt with acne scarring.

This is why it needs a careful, thought-out approach with targeted ingredients.

With over 30 years of dealing directly with the skin, we have found that the following three ingredients are the key to clear skin for many of our clients.

How to get rid of hyperpigmentation

3-O-Ethyl ascorbic acid 

Before proceeding, it’s important to mention that the form of vitamin C used is important for effectively treating deep-seated pigmentation.

Ascorbic acid can be unstable in specific formulations, so here at the Naked Chemist, we only ever formulate with 3-O-Ethyl ascorbic acid.

This is an ethylated form of vitamin C known for its stability and ability to penetrate the dermis (your skin’s deeper layers) to treat pigmentation.

This study (1), carried out over six months, found that participants who applied a cream-based lotion with just 5% 3-O-ethyl-l-ascorbic acid significantly improved their skin’s hyperpigmentation.

It was also observed that sunburn cell formation and inflammation signs were considerably reduced with regular application.

Human clinical trials (2) found it is very effective in treating hyperpigmentation due to its molecular size penetrating deep into the tyrosinase enzyme’s active site, disrupting copper ions and rendering the tyrosinase enzyme inactive.

A further study (3) found that repeated use of ethyl ascorbic acid scatters the pigment and lifts it out of the dermis, significantly helping to reduce melanin in the skin tissues.

3-O-Ethyl. Ascorbic acid also has numerous other benefits, such as boosting collagen synthesis, essential for maintaining your skin’s firmness and elasticity.

As we age, our bodies produce less collagen; therefore, regularly applying 3-O-Ethyl ascorbic acid can help to boost collagen production.

We love vitamin C so much that we have written extensively about it, which you can read here and here.

So, now that you understand how to get rid of hyperpigmentation with this primary ingredient, let’s explore the other two ingredients, which, when combined, form a powerful trio that can help you.

Age-defying ferulic acid

This clever ingredient works in synergy with 3-O-ethyl-l-ascorbic acid to combat pigmentation.

A potent antioxidant protects your skin from environmental aggressors like UV rays and pollution, which generate damaging free radicals.

Left unchecked, bothersome free radicals attack cell membranes and the mitochondria – the cell’s energy source – causing cellular damage and breaking down your skin’s healthy cells.

Antioxidant-rich ferulic acid neutralises these damaging free radicals, protecting your cells from oxidative stress that accelerates premature ageing.

Malic acid, the unsung hero

Malic acid is a powerful antioxidant and humectant with potent hydrating properties that place a protective, moisturising layer over your skin.

It works synergistically with ferulic and 3-O-ethyl-l-ascorbic acid to promote cellular turnover and reduce the skin’s rate of new pigment formation.

It is also an oil-loving hydroxy acid that helps reduce and slow down the oil flow in the sebaceous glands and unplugs stubborn debris that builds up in the pores, making it an excellent choice for oily, combination skin types.

A Beautiful Blend

So, how do you harness the benefits of these ingredients and know how to get rid hyperpigmentation for once and for all.?

Fortunately, we have synergistically combined them and put them together in one beautiful product, our C+ skin shot.

For best results, apply in the morning to take advantage of vitamin C and ferulic acid’s potent antioxidant properties.

There are some practical considerations that you should take into consideration when using this formula.

Start low and slow, especially if you have sensitive skin. We recommend initially using three times a week and slowly building your base. Once your skin builds up a tolerance, you can increase the usage.

We always recommend waiting 6 to 8 weeks of regular usage in line with cellular turnover before you can expect to see results.

If you are looking for other skin-lightening products from our range, our clients also get great results for treating deep-seated pigment issues layering with the following products:

Glo lactic acid skin shot,

A+ Retinol skin shot (Use at the opposite time of day to your C + skin shot).

Reset age delay cream (Use at the opposite time of day to your C+ skinshot).

To conclude. The naked truth

We have you covered if you want to know how to get rid of hyperpigmentation with specific ingredients.

Your hero ingredient should be vitamin C in the form of 3-O-ethyl-l-ascorbic acid combined with malic and ferulic acid.

Why? Because treating hyperpigmentation can be an extremely lengthy process, especially if it’s deep-seated.

This powerful trio works not only on the surface layers but also in the dermis (your deeper layer of skin) to remove dark spots, discolouration, and uneven skin tone, visibly improving luminosity, brightness, and texture.

And remember, consistency is the key in your journey to having radiant, clear skin.


1. Topical Vitamin C and the Skin: Mechanisms of Action and Clinical Applications

2. 3-O-ethyl-l-ascorbic acid: Characterisation and investigation of single solvent systems for delivery to the skin

3. The anti-melanogenic effects of 3-O-ethyl ascorbic acid via Nrf2-mediated α-MSH inhibition in UVA-irradiated keratinocytes and autophagy induction in melanocytes

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